| CBGA methyl ester | Olivetolic acid | ||
---|---|---|---|---|
(10 mg/kg, i.p.) | (10 mg/kg, i.p.) | |||
Plasma | Brain | Plasma | Brain | |
Cmax (μg/mL) | 1.3 ± 0.3 | 0.21 ± 0.03* | 65 ± 4 | 0.45 ± 0.06* |
tmax (min) | 45 | 30 | 15 | 15 |
t1/2 (min) | 81 | 62 | 10 | 14 |
AUC (μg•min/mL) | 171 | 22 | 1105 | 13 |
Brain-plasma ratio | 0.13 | 0.01 |